0 votes
15 views
ago in Chemical synthesis by (139k points)
What is the most efficient method to prepare 2-chloro-4-nitroaniline from aniline and chlorine gas while ensuring optimal yield and purity of the final product?

1 Answer

0 votes
ago by (139k points)
The most efficient method to prepare 2-chloro-4-nitroaniline from aniline and chlorine gas involves a two-step process:Step 1: Nitration of anilineFirst, you need to protect the amino group of aniline by acetylating it with acetic anhydride. This will form N-acetylaniline. The purpose of this step is to prevent the amino group from reacting with the nitration reagents in the next step.Next, nitrate the N-acetylaniline using a mixture of concentrated nitric acid  HNO3  and concentrated sulfuric acid  H2SO4 . This will form 4-nitro-N-acetylaniline.Step 2: ChlorinationIn this step, you will chlorinate the 4-nitro-N-acetylaniline. To do this, dissolve the 4-nitro-N-acetylaniline in an appropriate solvent, such as carbon tetrachloride  CCl4  or chloroform  CHCl3 . Then, bubble chlorine gas  Cl2  through the solution under controlled conditions  e.g., low temperature, controlled rate of Cl2 addition . This will form 2-chloro-4-nitro-N-acetylaniline.Finally, hydrolyze the 2-chloro-4-nitro-N-acetylaniline using aqueous hydrochloric acid  HCl  to remove the acetyl protecting group. This will yield the desired product, 2-chloro-4-nitroaniline.To ensure optimal yield and purity, it is crucial to monitor reaction conditions  e.g., temperature, concentration, and reaction time  and use appropriate purification techniques, such as recrystallization or column chromatography, after each step.

Related questions

Welcome to Sarvan Science Q&A, where you can ask questions and receive answers from other members of the community.
...